BDBM264086 2-[3-[1-(4- chlorophenyl)cyclopropyl]-5- hydroxypyrazol-1-yl]pyridine-4- carboxylic acid::US10173996, Example 171::US9604961, Example 171::US9714230, 171::US9908865, Example 171

SMILES OC(=O)c1ccnc(c1)-n1nc(cc1O)C1(CC1)c1ccc(Cl)cc1

InChI Key InChIKey=SCXPFBUUVUZXDW-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 264086   

TargetLysine-specific demethylase 2B(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 264086BDBM264086(2-[3-[1-(4- chlorophenyl)cyclopropyl]-5- hydroxypy...)
Affinity DataIC50: 100nMAssay Description:The ability of test compounds to inhibit the activity of FBXL10 was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details
US Patent

TargetLysine-specific demethylase 4C(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 264086BDBM264086(2-[3-[1-(4- chlorophenyl)cyclopropyl]-5- hydroxypy...)
Affinity DataIC50: 5.50E+3nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details
US Patent