BDBM270956 4-cyclopentyl-7-(4-methoxybenzenesulfonyl)-5H-pyrrolo[3,2-d]pyrimidin-6-amine::US10059713, Example 73

SMILES COc1ccc(cc1)S(=O)(=O)c1c(N)[nH]c2c(ncnc12)C1CCCC1

InChI Key InChIKey=SJUYXUIQTSTVLZ-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 270956   

TargetFree fatty acid receptor 2(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 270956BDBM270956(4-cyclopentyl-7-(4-methoxybenzenesulfonyl)-5H-pyrr...)
Affinity DataEC50:  9nMAssay Description:GPR43 agonist/PAM activity was determined by measuring changes in intracellular calcium levels using a Ca2+ sensitive fluorescent dye. The changes in...More data for this Ligand-Target Pair
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Date in BDB:
12/11/2018
Entry Details
US Patent