BDBM28803 2-[4-(4-chlorophenoxy)phenoxy]propanoic acid::Clofop::Fenofibric acid::HCG 004
SMILES CC(Oc1ccc(Oc2ccc(Cl)cc2)cc1)C(O)=O
InChI Key InChIKey=BSFAVVHPEZCASB-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 28803
Affinity DataIC50: >9.84E+4nM EC50: 1.16E+4nMpH: 8.0 T: 2°CAssay Description:For hPPAR alpha, percentage inhibition was calculated relative to unlabeled GW2331, which was used as the active site-specific competitive binder. Fl...More data for this Ligand-Target Pair
Affinity DataIC50: >9.84E+4nM EC50: >5.00E+4nMpH: 8.0 T: 2°CAssay Description:For PPARgamma, the percentage inhibition was calculated relative to rosiglitazone, which was used as the active site-specific competitive binder. Flu...More data for this Ligand-Target Pair
Affinity DataEC50: 1.77E+4nMAssay Description:EC50 is the concentration of test compounds needed to induce 50% of the maximum luciferase activity in HEK cells transfected with PPAR and Gal4-lucif...More data for this Ligand-Target Pair
Affinity DataEC50: 1.85E+4nMAssay Description:EC50 is the concentration of test compounds needed to induce 50% of the maximum luciferase activity in HEK cells transfected with PPAR and Gal4-lucif...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Mesocricetus auratus (golden hamster))
Bristol-Myers Squibb
Bristol-Myers Squibb
Affinity DataEC50: 2.87E+4nMAssay Description:EC50 is the concentration of test compounds needed to induce 50% of the maximum luciferase activity in HEK cells transfected with PPAR and Gal4-lucif...More data for this Ligand-Target Pair