BDBM365054 (R)-9-isobutyl-6,8-dimethyl- 4-(2-((1-methyl-1H-pyrazol- 5-yl)amino)pyrimidin-4-yl)- 8,9-dihydro-1,2,2a1,6,8- pentaazabenzo[cd]azulen- 7(6H)-one::US10278975, Compound I-19::US10517878, Compound I-19::US10842799, I-19::US11376260, Example I-19::US9867833, Compound I-19
SMILES CC(C)C[C@H]1N(C)C(=O)N(C)c2cc(cc3nnc1n23)-c1ccnc(Nc2ccnn2C)n1
InChI Key InChIKey=JFELDSBZJTUBGV-MRXNPFEDSA-N
Data 5 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 365054
Affinity DataIC50: 1.15nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: 1.15nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: 1.15nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: 1.15nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: 1.15nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair