BDBM365196 N-(1-methyl-1H-pyrazol-5- yl)-4-(9-(3,3,3- trifluoropropyl)-8,9-dihydro- 7H-6-oxa-1,2,2a1- triazabenzo[cd]azulen-4- yl)pyrimidin-2-amine::US10517878, Compound I-102::US10842799, I-102::US9867833, Compound I-102(S)
SMILES Cn1nccc1Nc1nccc(n1)-c1cc2OCCC(CCC(F)(F)F)c3nnc(c1)n23
InChI Key InChIKey=IZZPDFMHVSTMKH-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 365196
Affinity DataIC50: 0.0250nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair