BDBM469157 N-[6-(1,5-dimethyl-6-oxopyridin-3-yl)-1-[(4- fluorophenyl)methyl]-2-methylbenzimidazol-4- yl]methanesulfonamide::US10807982, Example 37
SMILES Cc1nc2c(NS(C)(=O)=O)cc(cc2n1Cc1ccc(F)cc1)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=KUEYACBOLWXVBE-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469157
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair