BDBM469174 N-[2-cyclopropyl-7-(1,5-dimethyl-6-oxopyridin- 3-yl)-3-methylbenzimidazol-5- yl]ethanesulfonamide::US10807982, Example 54
SMILES CCS(=O)(=O)Nc1cc(-c2cc(C)c(=O)n(C)c2)c2nc(C3CC3)n(C)c2c1
InChI Key InChIKey=FYJLBKZOWNHPPY-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469174
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair