BDBM469205 N-[4-(2,4-difluorophenoxy)-3-(6-methyl-5-oxo- 2,3-dihydro-1H-indolizin-8- yl)phenyl]methanesulfonamide::US10807982, Example 86
SMILES Cc1cc(c2CCCn2c1=O)-c1cc(NS(C)(=O)=O)ccc1Oc1ccc(F)cc1F
InChI Key InChIKey=PIUCATJBZCAYGQ-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469205
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair