BDBM469207 N-[4-(2,4-difluorophenoxy)-3-(2,2,6-trimethyl-5- oxo-1,3-dihydroindolizin-8- yl)phenyl]methanesulfonamide::US10807982, Example 88
SMILES Cc1cc(c2CC(C)(C)Cn2c1=O)-c1cc(NS(C)(=O)=O)ccc1Oc1ccc(F)cc1F
InChI Key InChIKey=GROYKANRBMYEOR-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469207
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair