BDBM469209 8-[2-(cyclopropylmethoxy)-5- methylsulfonylphenyl]-1-fluoro-6-methyl-2,3- dihydro-1H-indolizin-5-one::US10807982, Example 90
SMILES Cc1cc(c2C(F)CCn2c1=O)-c1cc(ccc1OCC1CC1)S(C)(=O)=O
InChI Key InChIKey=JOLCHACIXYRIRA-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469209
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair