BDBM469221 N-[5-(1,5-dimethyl-6-oxopyridin-3-yl)-3-[(4- fluorophenyl)methyl]-2-oxo-1,3-benzoxazol-7- yl]methanesulfonamide::US10807982, Example 102
SMILES Cc1cc(cn(C)c1=O)-c1cc(NS(C)(=O)=O)c2oc(=O)n(Cc3ccc(F)cc3)c2c1
InChI Key InChIKey=OBWZHFLXXDRKPG-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469221
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair