BDBM475045 US10849901, Compound 95::US10953012, Example 7
SMILES O=c1cc([nH]c2c(c(Cc3ccccc3)nn12)-c1ccccc1)-c1ccccc1
InChI Key InChIKey=SNTILYGOIGSXJU-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 475045
TargetPAS domain-containing serine/threonine-protein kinase [879-1323](Homo sapiens (Human))
Bioenergenix
US Patent
Bioenergenix
US Patent
Affinity DataIC50: >1.00E+4nMAssay Description:Table 1: One assay for purified hPASK activity utilizes the Kinase-Glo Luminescent Kinase Assay (Promega), which quantifies the amount of ATP remaini...More data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:The primary biochemical assay uses a fluorometric assay for monitoring the replacement of bound nucleotide with a fluorogenic GTP derivative bearing ...More data for this Ligand-Target Pair