BDBM476461 (2S)-4-{(4S,5S)-5-[3- (aminomethyl)phenyl]-4-methyl-4,5- dihydro-1,3-oxazol-2-yl}-1-[N2- cyclohexyl-N6-(methylsulfonyl)-D- lysyl]-N-(thiophen-2- ylmethyl)piperazine-2-carboxamide::US10875851, Example 117
SMILES C[C@@H]1N=C(O[C@H]1c1cccc(CN)c1)N1CCN([C@@H](C1)C(=O)NCc1cccs1)C(=O)[C@@H](CCCCNS(C)(=O)=O)NC1CCCCC1
InChI Key InChIKey=UXWDRYOJFUAWSY-QIXIFPRPSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 476461
Affinity DataIC50: 5.20nMAssay Description:The effectiveness of a compound of the present invention as an inhibitor of Coagulation Factor XIIa can be determined using a relevant purified serin...More data for this Ligand-Target Pair