BDBM476482 (2S)-4[(4S,5S)-5-(3-cyanophenyl)-4- methyl-4,5-dihydro-1,3-oxazol-2-yl]- 1-(N2-cyclohexyl-N6,N6-dimethyl-D- lysyl)-N-(thiophen-2- ylmethyl)piperazine-2-carboxamide::US10875851, Example 138
SMILES C[C@@H]1N=C(O[C@H]1c1cccc(c1)C#N)N1CCN([C@@H](C1)C(=O)NCc1cccs1)C(=O)[C@@H](CCCCN(C)C)NC1CCCCC1
InChI Key InChIKey=FKXSEWPZWBQOMC-QGWJVEIISA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 476482
Affinity DataIC50: 1.40nMAssay Description:The effectiveness of a compound of the present invention as an inhibitor of Coagulation Factor XIIa can be determined using a relevant purified serin...More data for this Ligand-Target Pair