BDBM481806 (R)-3-((6-chloro-2,3- dihydro-1H-inden-1- yl)methyl)-5-((7-methyl-6- oxo-6,7-dihydro-1H-purin- 1-yl)methyl-1,3,4-oxadiazol- 2(3H)-one::US10913742, Example 48
SMILES Cn1cnc2ncn(Cc3nn(C[C@@H]4CCc5ccc(Cl)cc45)c(=O)o3)c(=O)c12
InChI Key InChIKey=JYTFGJCBRILOIU-LBPRGKRZSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 481806
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 196nMAssay Description:The IC50 (effective concentration) of compounds on the human and rat TRPA1 channels were determined using a FLIPR Tetra instrument. CHO cells express...More data for this Ligand-Target Pair