BDBM481839 3-((4-((trans)-3-(4- chlorophenyl)cyclobutyl)-5- oxo-4,5-dihydro-1,3,4- oxadiazol-2-yl)methyl)-5- methylpyrido[3,2-d]pyrimidine- 4,6(3H,5H)-dione::US10913742, Example 83
SMILES Cn1c2c(ccc1=O)ncn(Cc1nn([C@H]3C[C@@H](C3)c3ccc(Cl)cc3)c(=O)o1)c2=O
InChI Key InChIKey=JOVMFRRSFHVPLP-CTYIDZIISA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 481839
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 15.2nMAssay Description:The IC50 (effective concentration) of compounds on the human and rat TRPA1 channels were determined using a FLIPR Tetra instrument. CHO cells express...More data for this Ligand-Target Pair