BDBM50130270 5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid ((S)-3-hexahydro-pyrrolo[1,2-a]pyrazin-2-yl-4-methoxy-phenyl)-amide::5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic acid [3-(hexahydro-pyrrolo[1,2-a]pyrazin-2-yl)-4-methoxy-phenyl]-amide::CHEMBL29433
SMILES COc1ccc(NS(=O)(=O)c2sc3ccc(Cl)cc3c2C)cc1N1CCN2CCC[C@H]2C1
InChI Key InChIKey=DVALOPXWVWHIHY-SFHVURJKSA-N
Data 17 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 17 hits for monomerid = 50130270
Affinity DataKi: 0.790nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.794nMAssay Description:The compound was tested for the binding affinity towards human cloned 5-hydroxytryptamine 6 receptor in HeLa cells, using [3H]5-LSD as radioligand; n...More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Antagonist activity at human recombinant 5HT6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity towards human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:The compound was tested for the binding affinity towards human cloned 5-hydroxytryptamine 1D receptor in CHO cells, using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:The compound was tested for the binding affinity towards human cloned 5-hydroxytryptamine 1A receptor in HEK293 cells, using [3H]8-OH-DPAT as radioli...More data for this Ligand-Target Pair
Affinity DataKi: 251nMAssay Description:The compound was tested for the binding affinity towards human cloned 5-hydroxytryptamine 2A receptor in HEK293 cells, using [3H]ketanserin as radiol...More data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:The compound was tested for the binding affinity towards human cloned 5-hydroxytryptamine 1F receptor in CHO cells, using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:The compound was tested for the binding affinity towards human cloned Dopamine receptor D3 in CHO cells, using [125I]iodosulpride as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:The compound was tested for the binding affinity towards human cloned 5-hydroxytryptamine 2C receptor in HEK293 cells, using [3H]5-mesulergine as rad...More data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:The compound was tested for the binding affinity towards human cloned 5-hydroxytryptamine 1B receptor in CHO cells, using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:The compound was tested for the binding affinity towards human cloned 5-hydroxytryptamine 7 receptor in HEK293 cells, using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+3nMAssay Description:The compound was tested for the binding affinity towards human cloned 5-hydroxytryptamine 2B receptor in HEK293 cells, using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.59E+3nMAssay Description:The compound was tested for the binding affinity towards human cloned 5-hydroxytryptamine 1E receptor in CHO cells, using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.59E+3nMAssay Description:The compound was tested for the binding affinity towards Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.59E+3nMAssay Description:The compound was tested for the binding affinity towards human cloned Dopamine receptor D2 in CHO cells, using [125I]iodosulpride as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5.01E+3nMAssay Description:The compound was tested for the binding affinity towards human cloned 5-hydroxytryptamine 4 receptor in HeLa cells, using [3H]LSD as radioligandMore data for this Ligand-Target Pair