BDBM50465300 CHEMBL4288985
SMILES COc1ccc(Br)cc1S(=O)(=O)Nc1ccc2NC(=O)C(C)(C)Oc2c1
InChI Key InChIKey=DZFJGVOWLQYSOW-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50465300
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Guangzhou Medical University
Curated by ChEMBL
Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.99E+3nMAssay Description:Inhibition of human His6-tagged BRD4 BD1 (N44 to E168 residues) expressed in Escherichia coli BL21 (DE3) cells using H-SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(A...More data for this Ligand-Target Pair