Affinity DataKi: 0.110nM ΔG°: -56.3kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.110nM ΔG°: -56.3kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: <0.25nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
Affinity DataKi: <0.25nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: <0.25nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.470nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 0.570nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.720nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 0.720nMAssay Description:Inhibition of chymotrypsin-like proteasome activity of human 20S proteasomeMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.940nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to FXa in presence of Zn2+More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to FXa in presence of Zn2+More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to thrombin in presence of Zn2+More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to factor7a/TF complexMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to FXa in presence of Zn2+More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human cathepsin BMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to F7a/TF complexMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to factor7a/TF complexMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to FXa in presence of Zn2+More data for this Ligand-Target Pair