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Found 36 with Last Name = 'taub' and Initial = 'd'
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50404997(CHEMBL18295)
Affinity DataIC50:  60nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50405004(CHEMBL282504)
Affinity DataIC50:  63nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50405001(CHEMBL273783)
Affinity DataIC50:  90nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50405003(CHEMBL428525)
Affinity DataIC50:  130nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50405007(CHEMBL18721)
Affinity DataIC50:  160nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50404998(CHEMBL276330)
Affinity DataIC50:  180nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50405002(CHEMBL19036)
Affinity DataIC50:  400nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50405010(CHEMBL18672)
Affinity DataIC50:  440nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50404999(CHEMBL282502)
Affinity DataIC50:  600nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50152559(4-Biphenyl-4-yl-2,4-dioxo-butyric acid | CHEMBL182...)
Affinity DataIC50:  1.10E+3nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50405005(CHEMBL279530)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50405000(CHEMBL18773)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50405009(CHEMBL19028)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50125793(4-(4-Cyclohexyl-phenyl)-2-hydroxy-4-oxo-but-2-enoi...)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022578(2-[(1-Amino-ethyl)-hydroxy-phosphinoylmethyl]-nona...)
Affinity DataIC50:  4.00E+3nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50367769(CHEMBL51843)
Affinity DataIC50:  4.00E+3nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022578(2-[(1-Amino-ethyl)-hydroxy-phosphinoylmethyl]-nona...)
Affinity DataIC50:  1.25E+4nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target2-Hydroxyacid oxidase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50405006(CHEMBL275811)
Affinity DataIC50:  1.90E+4nMAssay Description:In vitro inhibition of porcine Glycolate oxidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022569(2-[(1-Amino-ethyl)-hydroxy-phosphinoylmethyl]-pent...)
Affinity DataIC50:  2.00E+4nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022575(2-[(1-Amino-ethyl)-hydroxy-phosphinoylmethyl]-hexa...)
Affinity DataIC50:  2.00E+4nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022574(2-[(1-Amino-ethyl)-hydroxy-phosphinoylmethyl]-4-me...)
Affinity DataIC50:  3.00E+4nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50227637(CHEMBL3350233)
Affinity DataIC50:  3.50E+4nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022580(2-[(1-Amino-ethyl)-hydroxy-phosphinoylmethyl]-4-ph...)
Affinity DataIC50:  4.00E+4nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022577(2-[(1-Amino-ethyl)-hydroxy-phosphinoylmethyl]-buty...)
Affinity DataIC50:  4.50E+4nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM21459(3-[(1-aminoethyl)(hydroxy)phosphoryl]-2-benzylprop...)
Affinity DataIC50:  5.00E+4nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022579(2-[(1-Amino-ethyl)-hydroxy-phosphinoylmethyl]-5-ph...)
Affinity DataIC50:  5.00E+4nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022572(3-[(1-Amino-ethyl)-hydroxy-phosphinoyl]-2-methyl-p...)
Affinity DataIC50:  1.15E+5nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022573(2-[(1-Amino-propyl)-hydroxy-phosphinoylmethyl]-hex...)
Affinity DataIC50:  1.55E+5nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022572(3-[(1-Amino-ethyl)-hydroxy-phosphinoyl]-2-methyl-p...)
Affinity DataIC50:  1.65E+5nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022578(2-[(1-Amino-ethyl)-hydroxy-phosphinoylmethyl]-nona...)
Affinity DataIC50:  2.00E+5nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50014155(CHEMBL3260854)
Affinity DataIC50:  2.15E+5nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50038178((+)-4-Amino-3-isoxazolidinone | (4R)-4-aminoisoxaz...)
Affinity DataIC50:  3.00E+5nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022576(3-[(1-Amino-ethyl)-hydroxy-phosphinoyl]-propionic ...)
Affinity DataIC50:  5.35E+5nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50017377((1-Amino-ethyl)-phosphonic acid | 1-Ammonium-ethan...)
Affinity DataIC50:  9.30E+5nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022571(CHEMBL299420 | D-Ala-D-Ala | D-alanyl-D-alanine)
Affinity DataIC50:  1.00E+6nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligase(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50022570(1-aminoethylphosphonous acid | CHEMBL300051)
Affinity DataIC50:  1.00E+6nMAssay Description:Antibacterial activity against D-alanyl-D-alanine ligase from Streptococcus faecalis (ATCC 8043)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed