TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego
Curated by ChEMBL
University Of California San Diego
Curated by ChEMBL
Affinity DataIC50: 0.0200nMAssay Description:Inhibitory concentration against human somatostatin receptor type 2 in CC531 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor mSSTR2bMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego
Curated by ChEMBL
University Of California San Diego
Curated by ChEMBL
Affinity DataIC50: 0.770nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor hSSTR5More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor rSSTR5More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor mSSTR3More data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of California San Diego
Curated by ChEMBL
University Of California San Diego
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor hSSTR4More data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego
Curated by ChEMBL
University Of California San Diego
Curated by ChEMBL
Affinity DataIC50: 21.8nMAssay Description:Inhibitory concentration against human somatostatin receptor type 5 in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego
Curated by ChEMBL
University Of California San Diego
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human SSTR5 by radioligand binding assayMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego
Curated by ChEMBL
University Of California San Diego
Curated by ChEMBL
Affinity DataIC50: 92.9nMAssay Description:Inhibitory concentration against human somatostatin receptor type 3 in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of California San Diego
Curated by ChEMBL
University Of California San Diego
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human SSTR4 by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.34E+3nMAssay Description:Inhibition of human BSEP overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-taurocholate in presence of ATP measured after 15 to ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.33E+5nMAssay Description:Inhibition of human MRP2 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...More data for this Ligand-Target Pair
Affinity DataIC50: >1.33E+5nMAssay Description:Inhibition of human MRP4 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...More data for this Ligand-Target Pair
Affinity DataIC50: >1.33E+5nMAssay Description:Inhibition of human MRP3 overexpressed in Sf9 insect cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ...More data for this Ligand-Target Pair