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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A' and Ligand = 'BDBM50316678'
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316678(8-{4-[4-(6-Methoxyquinolin-8-yl)piperazin-1-yl]pip...)
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316678(8-{4-[4-(6-Methoxyquinolin-8-yl)piperazin-1-yl]pip...)
Affinity DataIC50:  4.80nMAssay Description:Antagonist activity at human 5HT1A receptor expressed in CHO cells assessed as blockade of 8-OH-DPAT-induced inhibition of forskolin-stimulated incre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed