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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2b' and Ligand = 'BDBM50025585'
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50025585(7-(2-Hydroxy-ethyl)-1,3-dimethyl-3,7-dihydro-purin...)
Affinity DataKi:  1.73E+4nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50025585(7-(2-Hydroxy-ethyl)-1,3-dimethyl-3,7-dihydro-purin...)
Affinity DataKi:  1.73E+4nMAssay Description:Binding affinity at human Adenosine A2B receptor expressed in HEK-293 cells, using [125I]-ABOPX as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed