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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2b' and Ligand = 'BDBM50150077'
TargetAdenosine receptor A2b(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50150077(2-((1H-imidazol-2-yl)methylthio)-6-amino-4-phenylp...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]PSB-603 from human A2B receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50150077(2-((1H-imidazol-2-yl)methylthio)-6-amino-4-phenylp...)
Affinity DataEC50:  19nMAssay Description:Agonistic activity against human adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed