Affinity DataKi: 160nMAssay Description:The compound was evaluated for the binding affinity towards Dopamine receptor D2 at high affinity stateMore data for this Ligand-Target Pair
Affinity DataKi: 6.87E+3nMAssay Description:Binding affinity was determined by measuring the ability to displace [125I]N-(p-aminophenethyl)-spiroperidol from Dopamine receptor D2 in rat caudate...More data for this Ligand-Target Pair
Affinity DataKi: 6.87E+3nMAssay Description:Binding affinity was determined by measuring the ability to displace [125I]N-(p-aminophenethyl)-spiroperidol from Dopamine receptor D2 in rat caudate...More data for this Ligand-Target Pair
Affinity DataKi: 8.80E+3nMAssay Description:The compound was evaluated for the binding affinity towards Dopamine receptor D2 at low affinity stateMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20E+5nMAssay Description:Displacement of [3H]-YM-09151-2 (60 pm) from dopamine receptor D2 in crude membrane fraction of rat brain corpus striatumMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Formation of cAMP on Dopamine receptor D2 in vitro in rat intermediate lobeMore data for this Ligand-Target Pair
Affinity DataKd: 1.35E+5nMAssay Description:In vitro affinity at mutant D2 receptor (S197A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
Affinity DataKd: 4.60E+4nMAssay Description:In vitro affinity at wild type Dopamine receptor D2 on C6 (glioma) cell membranes.More data for this Ligand-Target Pair
Affinity DataKd: 1.80E+4nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
Affinity DataKd: 3.90E+4nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair