TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 0.220nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at human mu opioid receptor expressed in human U2OS cells co-transfected with beta-arrestin-2 assessed as increase in beta-arrestin-...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
Affinity DataEC50: 1.30nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cell membranes after 1 hr by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair