Found 3 Enz. Inhib. hit(s) with Target = 'Solute carrier family 22 member 8' and Ligand = 'BDBM50022787'
Affinity DataKi: 5.28E+4nMAssay Description:TP_TRANSPORTER: inhibition of Pravastatin uptake in Oat3-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.76E+4nMAssay Description:TP_TRANSPORTER: inhibition of MTX uptake in OAT3-expressing S2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.94E+4nMAssay Description:Inhibition of mouse OAT3 expressed in CHO cells assessed as inhibition of fluorescein uptake over 20 minsMore data for this Ligand-Target Pair