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Found 1 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK1' and Ligand = 'BDBM466937'
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466937(US10800775, Example 17 | ethyl 4-(1-(2-cyano-1-cyc...)
Affinity DataIC50:  55nMAssay Description:The activity of JAK3 (a.a. 781-1124, ThermoFisher) was quantified by measuring the phosphorylation of SRCtide (FAM-GEEPLYWSFPAKKK-NH2). Kinase reacti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent