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Found
1
Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK1' and Ligand = 'BDBM475719'
Target
Tyrosine-protein kinase JAK1
(Homo sapiens (Human))
Leo Pharma
US Patent
Ligand
BDBM475719
(2-[(3aS*,7aS*)-3a-methyl-5-(7H-pyrrolo[2,3-d]pyrim...)
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Affinity Data
EC50: 49nM
Assay Description:
Inhibition of phosphorylation of a synthetic peptide was measured in an HTRF-based assay using the TK substrate-Biotin from the Cisbio HTRFKinEASE TK...
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Target Info
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Ligand Info
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Details
US Patent
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