Affinity DataEC50: 30nMAssay Description:Inhibition of HDAC in human cell lysates using fluoro-substrate peptide/fluoro-deacetylated peptide as substrate incubated for 20 mins measured at 1 ...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
S£O Paulo State University (Unesp)
Curated by ChEMBL
S£O Paulo State University (Unesp)
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Inhibition of recombinant human HDAC1 expressed in baculovirus expression system using KI-104 as substrate incubated for 3 hrs by by fluorescence-bas...More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
S£O Paulo State University (Unesp)
Curated by ChEMBL
S£O Paulo State University (Unesp)
Curated by ChEMBL
Affinity DataEC50: 125nMAssay Description:Inhibition of recombinant human HDAC2 expressed in baculovirus expression system using KI-104 as substrate incubated for 3 hrs by by fluorescence-bas...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
S£O Paulo State University (Unesp)
Curated by ChEMBL
S£O Paulo State University (Unesp)
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Inhibition of recombinant human HDAC3 expressed in baculovirus expression system using KI-104 as substrate incubated for 3 hrs by by fluorescence-bas...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
S£O Paulo State University (Unesp)
Curated by ChEMBL
S£O Paulo State University (Unesp)
Curated by ChEMBL
Affinity DataEC50: 216nMAssay Description:Inhibition of recombinant human HDAC8 expressed in baculovirus expression system using FDL as substrate incubated for 3 hrs by by fluorescence-based ...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
S£O Paulo State University (Unesp)
Curated by ChEMBL
S£O Paulo State University (Unesp)
Curated by ChEMBL
Affinity DataEC50: 82nMAssay Description:Inhibition of recombinant human HDAC6 expressed in baculovirus expression system using KI-104 as substrate incubated for 3 hrs by by fluorescence-bas...More data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
S£O Paulo State University (Unesp)
Curated by ChEMBL
S£O Paulo State University (Unesp)
Curated by ChEMBL
Affinity DataEC50: 67nMAssay Description:Inhibition of recombinant human HDAC7 expressed in baculovirus expression system using KI-104 as substrate incubated for 3 hrs by by fluorescence-bas...More data for this Ligand-Target Pair
TargetHistone deacetylase 9(Homo sapiens (Human))
S£O Paulo State University (Unesp)
Curated by ChEMBL
S£O Paulo State University (Unesp)
Curated by ChEMBL
Affinity DataEC50: 128nMAssay Description:Inhibition of recombinant human HDAC9 expressed in baculovirus expression system using KI-104 as substrate incubated for 3 hrs by by fluorescence-bas...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
S£O Paulo State University (Unesp)
Curated by ChEMBL
S£O Paulo State University (Unesp)
Curated by ChEMBL
Affinity DataEC50: 115nMAssay Description:Inhibition of recombinant human HDAC4 expressed in baculovirus expression system using KI-104 as substrate incubated for 3 hrs by by fluorescence-bas...More data for this Ligand-Target Pair