Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for UniProtKB: Q63424
TargetSolute carrier family 15 member 2(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50344967(2-[(4-Isopropyl-cyclohexanecarbonyl)-amino]-3-phen...)
Affinity DataIC50:  7.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 20 uM) in PEPT2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 2(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM17658((2S)-2-[(3S)-3-acetamido-3-formamidopropanoic acid...)
Affinity DataIC50:  3.00E+6nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 10 uM) in PEPT2-expressing SK-N-SH cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 2(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM84007(CEFIXIME | Cefiximum [Latin] | MLS002222332 | SMR0...)
Affinity DataIC50:  3.20E+6nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 5 uM) in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 2(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50248190(CHEBI:3485 | CI-983 | Cefdinir | Cefzon | FK-482 |...)
Affinity DataIC50:  1.00E+7nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 5 uM) in SKPT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed