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Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50001852
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  31nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50:  74nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50:  98nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50:  270nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50:  290nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50:  740nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50:  760nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50:  1.67E+3nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human CDK2/CyclinA using histone H1 as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406884(CHEMBL4168687)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human CDK2/CyclinA using histone H1 as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT expressed in baculovirus infected Sf9 insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) expressed in bacterial expression system using histone H3 peptide as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacterial expression system using GRSRSRSRSRSR as substrate after 30 mins by ADP-Glo reagent based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Sus scrofa)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406885(CHEMBL4170635)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Sus scrofa)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) expressed in bacterial expression system using histone H3 peptide as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT expressed in baculovirus infected Sf9 insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406886(CHEMBL4169579)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Sus scrofa)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406887(CHEMBL4162709)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406888(CHEMBL4175950)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406889(CHEMBL4168098)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406890(CHEMBL4173649)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human CDK2/CyclinA using histone H1 as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT expressed in baculovirus infected Sf9 insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) expressed in bacterial expression system using histone H3 peptide as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacterial expression system using GRSRSRSRSRSR as substrate after 30 mins by ADP-Glo reagent based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Sus scrofa)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406891(CHEMBL4163110)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406892(CHEMBL4159749)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406989(CHEMBL4162053)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50407008(CHEMBL4170051)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT expressed in baculovirus infected Sf9 insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) expressed in bacterial expression system using histone H3 peptide as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT expressed in baculovirus infected Sf9 insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human haspin kinase domain (470 to 798 residues) expressed in bacterial expression system using histone H3 peptide as subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacterial expression system using GRSRSRSRSRSR as substrate after 30 mins by ADP-Glo reagent based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta/[Tau protein] kinase(Sus scrofa)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406883(CHEMBL4177432)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of porcine brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human CDK2/CyclinA using histone H1 as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406881(CHEMBL4177174)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406880(CHEMBL4170384)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human CDK2/CyclinA using histone H1 as substrate after 30 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406882(CHEMBL4166554)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacterial expression system using GRSRSRSRSRSR as substrate after 30 mins by ADP-Glo reagent based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406878(CHEMBL4166150)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Pim1 expressed in bacterial expression system using histone H1 as substrate after 30 mins by ADP-Glo reagent based lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mus musculus)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50406879(CHEMBL4174068)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacterial expression system using GRSRSRSRSRSR as substrate after 30 mins by ADP-Glo reagent based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed