Compile Data Set for Download or QSAR
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Report error Found 138 Enz. Inhib. hit(s) with all data for entry = 50009606
TargetD(4) dopamine receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50530438(Mosapramine | Mosapramine hydrochloride)
Affinity DataKi:  0.0300nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50530438(Mosapramine | Mosapramine hydrochloride)
Affinity DataKi:  0.0300nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50274351(2-(6,8-Dichloro-2-(4-nitrophenyl)imidazo[1,2-a]pyr...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50274351(2-(6,8-Dichloro-2-(4-nitrophenyl)imidazo[1,2-a]pyr...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
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Curated by ChEMBL
LigandPNGBDBM50247053(1-(3-(3-(4-chlorophenyl)propoxy)propyl)piperidine ...)
Affinity DataKi:  0.160nMAssay Description:Inhibition of Guinea Pig Ileum H3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
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Curated by ChEMBL
LigandPNGBDBM50247053(1-(3-(3-(4-chlorophenyl)propoxy)propyl)piperidine ...)
Affinity DataKi:  0.160nMAssay Description:Inhibition of Guinea Pig Ileum H3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50189854(6-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  0.25nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50189854(6-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  0.25nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50189841(6-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataKi:  0.330nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50189841(6-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataKi:  0.330nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50060095(2-[6,8-Dichloro-2-(4-chloro-phenyl)-imidazo[1,2-a]...)
Affinity DataKi:  0.410nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50060095(2-[6,8-Dichloro-2-(4-chloro-phenyl)-imidazo[1,2-a]...)
Affinity DataKi:  0.410nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50530421(CHEMBL4585201)
Affinity DataKi:  0.5nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50530421(CHEMBL4585201)
Affinity DataKi:  0.5nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50274258(2-(6,8-Dichloro-2-(4-methoxyphenyl)imidazo[1,2-a]p...)
Affinity DataKi:  0.537nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50274258(2-(6,8-Dichloro-2-(4-methoxyphenyl)imidazo[1,2-a]p...)
Affinity DataKi:  0.537nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50530440(CHEMBL4548796)
Affinity DataKi:  0.75nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50530440(CHEMBL4548796)
Affinity DataKi:  0.75nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50274561(4-(2-(4-Chlorophenyl)-3-(2-(dipropylamino)-2-oxoet...)
Affinity DataKi:  0.860nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50274561(4-(2-(4-Chlorophenyl)-3-(2-(dipropylamino)-2-oxoet...)
Affinity DataKi:  0.860nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50274259(CHEMBL521186 | N-Butyl-2-(6,8-dichloro-2-(4-methox...)
Affinity DataKi:  0.882nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50274259(CHEMBL521186 | N-Butyl-2-(6,8-dichloro-2-(4-methox...)
Affinity DataKi:  0.882nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50189848(2-[4-(3,4-dichlorophenyl)piperazin-1-ylmethyl]imid...)
Affinity DataKi:  0.990nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50189848(2-[4-(3,4-dichlorophenyl)piperazin-1-ylmethyl]imid...)
Affinity DataKi:  0.990nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50408728(CHEMBL339816)
Affinity DataKi:  1.60nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50408728(CHEMBL339816)
Affinity DataKi:  1.60nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50120543(7-Methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)
Affinity DataKi:  2nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50120543(7-Methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)
Affinity DataKi:  2nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50530442(CHEMBL4461114)
Affinity DataKi:  2.10nMAssay Description:Inhibition of human PDE10More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50530442(CHEMBL4461114)
Affinity DataKi:  2.10nMAssay Description:Inhibition of human PDE10More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50189845(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo...)
Affinity DataKi:  2.80nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50189845(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo...)
Affinity DataKi:  2.80nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50045880(2-[5-Chloro-2-(4-chloro-phenyl)-1H-indol-3-yl]-N,N...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50045880(2-[5-Chloro-2-(4-chloro-phenyl)-1H-indol-3-yl]-N,N...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50189842(2-[4-(4-chlorophenyl)piperazin-1-yl)methyl]imidazo...)
Affinity DataKi:  7nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50189842(2-[4-(4-chlorophenyl)piperazin-1-yl)methyl]imidazo...)
Affinity DataKi:  7nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50530422(CHEMBL4468363)
Affinity DataKi:  12nMAssay Description:Antagonist activity at 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50011297(CHEMBL3260729 | US9029393, 14)
Affinity DataKi:  12nMAssay Description:Inhibition of GFP-tagged human A2A adenosine receptor expressed in HEK cells by FRET-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50530422(CHEMBL4468363)
Affinity DataKi:  12nMAssay Description:Antagonist activity at 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Palack£

Curated by ChEMBL
LigandPNGBDBM159248(US9034874, 1.5)
Affinity DataKi:  12nMAssay Description:Inhibition of Guinea Pig Ileum H3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Palack£

Curated by ChEMBL
LigandPNGBDBM159248(US9034874, 1.5)
Affinity DataKi:  12nMAssay Description:Inhibition of Guinea Pig Ileum H3RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50011297(CHEMBL3260729 | US9029393, 14)
Affinity DataKi:  12nMAssay Description:Inhibition of GFP-tagged human A2A adenosine receptor expressed in HEK cells by FRET-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50530420(CHEMBL4450928)
Affinity DataKi:  14nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50530420(CHEMBL4450928)
Affinity DataKi:  14nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM26266(Ambien | CHEMBL911 | Dalparan | N,N-dimethyl-2-[6-...)
Affinity DataKi:  20nMAssay Description:Inhibition of GABAA receptor alpha1 (unknown origin)More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM26266(Ambien | CHEMBL911 | Dalparan | N,N-dimethyl-2-[6-...)
Affinity DataKi:  20nMAssay Description:Inhibition of GABAA receptor alpha1 (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50530424(CHEMBL4533922)
Affinity DataKi:  26nMAssay Description:Antagonist activity at 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50530424(CHEMBL4533922)
Affinity DataKi:  26nMAssay Description:Antagonist activity at 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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