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Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50014268
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  30nMAssay Description:Inhibition of PIM1 (unknown origin) in presence of 1 mM ATP without preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  34nMAssay Description:Inhibition of PIM1 (unknown origin) in presence of 1 mM ATP with preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  36nMAssay Description:Inhibition of CDC7 in human SW-620 cells assessed as reduction in phosphorylation of MCM2 at Ser40 residue incubated for 48 hrs by Western blot analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  53nMAssay Description:Inhibition of CDC7 in human SW-620 cells assessed as reduction in phosphorylation of MCM2 at Ser53 residue incubated for 48 hrs by Western blot analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  189nMAssay Description:Inhibition of GSK3alpha (unknown origin) in presence of 1 mM ATP without preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  206nMAssay Description:Inhibition of CLK1 (unknown origin) in presence of 1 mM ATP with preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  212nMAssay Description:Inhibition of CLK1 (unknown origin) in presence of 1 mM ATP without preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  227nMAssay Description:Inhibition of CLK2 (unknown origin) in presence of 1 mM ATP with preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  251nMAssay Description:Inhibition of GSK3alpha (unknown origin) in presence of 1 mM ATP with preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  270nMAssay Description:Inhibition of CLK2 (unknown origin) in presence of 1 mM ATP without preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed