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Report error Found 90 Enz. Inhib. hit(s) with all data for entry = 50029707
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287090(4-Chloro-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2...)
Affinity DataIC50:  10nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50175491(4-Methyl-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2...)
Affinity DataIC50:  10nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287091(CHEMBL20252 | Naphthalene-2-carboxylic acid [4-met...)
Affinity DataIC50:  50nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240407(CHEMBL20926 | N-(4-methyl-3-(4-(pyridin-3-yl)pyrim...)
Affinity DataIC50:  100nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287094(CHEMBL278630 | N-[4-Chloro-3-(4-pyridin-3-yl-pyrim...)
Affinity DataIC50:  150nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287096(2-Methoxy-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50175493(CHEMBL277931 | N-[3-(4-Pyridin-3-yl-pyrimidin-2-yl...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287092(CHEMBL277430 | N-Benzoyl-N-[4-methyl-3-(4-pyridin-...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50175493(CHEMBL277931 | N-[3-(4-Pyridin-3-yl-pyrimidin-2-yl...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287087(CHEMBL21078 | N-[4-Methyl-3-(4-thiophen-2-yl-pyrim...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287095(4,N*1*-Dimethyl-N*3*-(4-pyridin-3-yl-pyrimidin-2-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287097(4-Methyl-N*3*-(4-pyridin-3-yl-pyrimidin-2-yl)-benz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287088(CHEMBL21086 | N-[4-Methoxy-3-(4-pyridin-3-yl-pyrim...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287098(CHEMBL21079 | N-{4-Methyl-3-[4-(1-oxy-pyridin-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287088(CHEMBL21086 | N-[4-Methoxy-3-(4-pyridin-3-yl-pyrim...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50175493(CHEMBL277931 | N-[3-(4-Pyridin-3-yl-pyrimidin-2-yl...)
Affinity DataIC50:  1.57E+4nMAssay Description:Inhibition of tyrosine kinase(c-Src)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C delta type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50175493(CHEMBL277931 | N-[3-(4-Pyridin-3-yl-pyrimidin-2-yl...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of serine/threonine kinase(PKC-delta)More data for this Ligand-Target Pair
In DepthDetails Article
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287089(CHEMBL278287 | N-Methyl-N-[4-methyl-3-(4-pyridin-3...)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of tyrosine kinase Epidermal growth factor receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50175493(CHEMBL277931 | N-[3-(4-Pyridin-3-yl-pyrimidin-2-yl...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of tyrosine kinase Epidermal growth factor receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240406(CHEMBL423288 | N-(4-methyl-3-(4-(pyridin-3-yl)pyri...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287095(4,N*1*-Dimethyl-N*3*-(4-pyridin-3-yl-pyrimidin-2-y...)
Affinity DataIC50:  7.10E+4nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240407(CHEMBL20926 | N-(4-methyl-3-(4-(pyridin-3-yl)pyrim...)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287092(CHEMBL277430 | N-Benzoyl-N-[4-methyl-3-(4-pyridin-...)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibition of tyrosine kinase Epidermal growth factor receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287089(CHEMBL278287 | N-Methyl-N-[4-methyl-3-(4-pyridin-3...)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287091(CHEMBL20252 | Naphthalene-2-carboxylic acid [4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287096(2-Methoxy-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287092(CHEMBL277430 | N-Benzoyl-N-[4-methyl-3-(4-pyridin-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240406(CHEMBL423288 | N-(4-methyl-3-(4-(pyridin-3-yl)pyri...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287090(4-Chloro-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287087(CHEMBL21078 | N-[4-Methyl-3-(4-thiophen-2-yl-pyrim...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287094(CHEMBL278630 | N-[4-Chloro-3-(4-pyridin-3-yl-pyrim...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50175491(4-Methyl-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287098(CHEMBL21079 | N-{4-Methyl-3-[4-(1-oxy-pyridin-3-yl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287097(4-Methyl-N*3*-(4-pyridin-3-yl-pyrimidin-2-yl)-benz...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-alpha)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C delta type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287089(CHEMBL278287 | N-Methyl-N-[4-methyl-3-(4-pyridin-3...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-delta)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C delta type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287098(CHEMBL21079 | N-{4-Methyl-3-[4-(1-oxy-pyridin-3-yl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-delta)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287096(2-Methoxy-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of tyrosine kinase(c-Src)More data for this Ligand-Target Pair
In DepthDetails Article
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287094(CHEMBL278630 | N-[4-Chloro-3-(4-pyridin-3-yl-pyrim...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of tyrosine kinase Epidermal growth factor receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287090(4-Chloro-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of tyrosine kinase(c-Src)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240407(CHEMBL20926 | N-(4-methyl-3-(4-(pyridin-3-yl)pyrim...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of tyrosine kinase(c-Src)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287093((2-Methyl-5-nitro-phenyl)-(4-pyridin-3-yl-pyrimidi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of tyrosine kinase(c-Src)More data for this Ligand-Target Pair
In DepthDetails Article
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287098(CHEMBL21079 | N-{4-Methyl-3-[4-(1-oxy-pyridin-3-yl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of tyrosine kinase Epidermal growth factor receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240407(CHEMBL20926 | N-(4-methyl-3-(4-(pyridin-3-yl)pyrim...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of tyrosine kinase Epidermal growth factor receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C delta type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287092(CHEMBL277430 | N-Benzoyl-N-[4-methyl-3-(4-pyridin-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-delta)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C delta type(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287088(CHEMBL21086 | N-[4-Methoxy-3-(4-pyridin-3-yl-pyrim...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKC-delta)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287089(CHEMBL278287 | N-Methyl-N-[4-methyl-3-(4-pyridin-3...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287093((2-Methyl-5-nitro-phenyl)-(4-pyridin-3-yl-pyrimidi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287091(CHEMBL20252 | Naphthalene-2-carboxylic acid [4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of tyrosine kinase(PDGF-R)More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50175491(4-Methyl-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKA)More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287090(4-Chloro-N-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of serine/threonine kinase(PKA)More data for this Ligand-Target Pair
In DepthDetails Article
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