Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 50037865
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196700(5-((3-(3-(prop-1-en-2-yl)benzyl)cyclohexyl)methyl)...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196694(CHEMBL225166 | N-(1-(thiophen-3-ylmethyl)piperidin...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196718(CHEMBL373512 | N-(1-(thiophen-2-ylmethyl)piperidin...)
Affinity DataIC50:  5nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196692(CHEMBL388516 | N-(1-(4-methylbenzyl)piperidin-3-yl...)
Affinity DataIC50:  9nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196695(CHEMBL224510 | N-(1-(3,4-difluorobenzyl)piperidin-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196711(1-benzyl-3-piperidyl-(1H-5-indazolyl)ether | 5-(1-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196690(CHEMBL224535 | N-(1-(4-aminobenzyl)piperidin-3-yl)...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196689(CHEMBL224166 | N-(1-((1H-pyrrol-2-yl)methyl)piperi...)
Affinity DataIC50:  11nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196682(CHEMBL426925 | N-(1-(4-chlorobenzyl)piperidin-3-yl...)
Affinity DataIC50:  11nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196707(CHEMBL390837 | N-(1-(2-chlorobenzyl)piperidin-3-yl...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196712(CHEMBL225637 | N-(1-(4-methoxybenzyl)piperidin-3-y...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196704(1-benzyl-N-(1H-5-indazolyl)piperidine-3-carboxamid...)
Affinity DataIC50:  18nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196728(CHEMBL389168 | N-(1-(3-chlorobenzyl)piperidin-3-yl...)
Affinity DataIC50:  19nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196698(CHEMBL390389 | N-(1-(3-chlorobenzyl)pyrrolidin-3-y...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196725(CHEMBL224885 | N-(1-benzyl-3-piperidyl)-N-(1H-5-in...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196725(CHEMBL224885 | N-(1-benzyl-3-piperidyl)-N-(1H-5-in...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196687(1-(2,6-dichlorobenzyl)-3-(1H-indazol-5-yl)urea | 1...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196686(CHEMBL427245 | N-(1-(4-chlorobenzyl)pyrrolidin-3-y...)
Affinity DataIC50:  24nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196688(CHEMBL224509 | N-(1-(4-fluorobenzyl)piperidin-3-yl...)
Affinity DataIC50:  25nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196708(CHEMBL386937 | N-(1-benzyl-3-pyrrolidyl)-N-(1H-5-i...)
Affinity DataIC50:  32nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196699(CHEMBL390736 | N-(1-(3-aminobenzyl)piperidin-3-yl)...)
Affinity DataIC50:  35nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196679(CHEMBL388742 | N-(1-(2-chlorobenzyl)pyrrolidin-3-y...)
Affinity DataIC50:  45nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196706(CHEMBL225167 | N-(1-(furan-2-ylmethyl)piperidin-3-...)
Affinity DataIC50:  65nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196683(CHEMBL224746 | N-(1-(pyridin-3-ylmethyl)piperidin-...)
Affinity DataIC50:  72nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196685(CHEMBL389622 | N-(1-(3,5-dimethoxybenzyl)piperidin...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196702(CHEMBL427254 | N-(1-(2-aminobenzyl)piperidin-3-yl)...)
Affinity DataIC50:  85nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196681(1-(2,6-difluorobenzyl)-3-(1H-indazol-5-yl)urea | C...)
Affinity DataIC50:  85nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196691(CHEMBL389915 | N-(1-(4-nitrobenzyl)piperidin-3-yl)...)
Affinity DataIC50:  87nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196696(1-benzyl-4-piperidyl-(1H-5-indazolyl)ether | 5-(1-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196684(1-benzyl-N-(1H-5-indazolyl)piperidine-4-carboxamid...)
Affinity DataIC50:  136nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM107898(CHEMBL373487 | US8604218, 1.049)
Affinity DataIC50:  150nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM14027(5-(1,4-diazepan-1-ylsulfonyl)isoquinoline | 5-(1,4...)
Affinity DataIC50:  180nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196720(CHEMBL225168 | N-[1-(3-furylmethyl)-3-piperidyl]-N...)
Affinity DataIC50:  180nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196701(CHEMBL224533 | N-(1-(pyridin-4-ylmethyl)piperidin-...)
Affinity DataIC50:  190nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196709(1-(2,4-dichlorobenzyl)-3-(1H-indazol-5-yl)urea | C...)
Affinity DataIC50:  220nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196721(CHEMBL224696 | N-(1-(pyridin-2-ylmethyl)piperidin-...)
Affinity DataIC50:  240nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196680(CHEMBL224500 | N-(1-benzyl-4-piperidyl)-N-(1H-5-in...)
Affinity DataIC50:  240nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196697(1-benzyl-3-(1H-indazol-5-yl)urea | CHEMBL225282 | ...)
Affinity DataIC50:  260nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196723(CHEMBL225225 | N-(1-(4-chlorobenzyl)piperidin-4-yl...)
Affinity DataIC50:  290nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196719(CHEMBL224559 | N-(1-(3-chlorobenzyl)piperidin-4-yl...)
Affinity DataIC50:  290nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196716(CHEMBL390390 | N1-benzyl-N4-(1H-5-indazolyl)-1,4-c...)
Affinity DataIC50:  320nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196722(CHEMBL427085 | N-(1-isobutylpiperidin-3-yl)-1H-ind...)
Affinity DataIC50:  340nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196727(CHEMBL224558 | N-(1-(2-chlorobenzyl)piperidin-4-yl...)
Affinity DataIC50:  440nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196715(CHEMBL224067 | N1-benzyl-N4-(1H-5-indazolyl)-1,4-c...)
Affinity DataIC50:  520nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196705(CHEMBL223651 | N-(1-benzylpiperidin-4-yl)-1H-indaz...)
Affinity DataIC50:  540nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196703(CHEMBL223553 | N-(1-ethylpiperidin-3-yl)-1H-indazo...)
Affinity DataIC50:  780nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196712(CHEMBL225637 | N-(1-(4-methoxybenzyl)piperidin-3-y...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of MCP1-induced cell migration in U937 cells expressing CCR2 by chemotaxis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 1/2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196710(CHEMBL224167 | N-[1-(1H-3-pyrrolylmethyl)-3-piperi...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of Rho kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196695(CHEMBL224510 | N-(1-(3,4-difluorobenzyl)piperidin-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of MCP1-induced cell migration in U937 cells expressing CCR2 by chemotaxis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Kirin Brewery

Curated by ChEMBL
LigandPNGBDBM50196692(CHEMBL388516 | N-(1-(4-methylbenzyl)piperidin-3-yl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of MCP1-induced cell migration in U937 cells expressing CCR2 by chemotaxis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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