Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50044699
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant LRRK2 G2019S mutant (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiog...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant GSK3alpha using CFFKNIVTPRTPPPSQGK-amide substrate after 60 mins incubation by LANCE methodMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant GSK3beta using CFFKNIVTPRTPPPSQGK-amide substrate after 90 mins incubation by LANCE methodMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of recombinant LRRK2 G2019S mutant (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiog...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 163nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 194nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 204nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 205nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 261nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 466nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Technische Universit£T Darmstadt
Curated by ChEMBL
Technische Universit£T Darmstadt
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of recombinant LRRK2 (unknown origin) using gamma-32P-ATP assessed as LRRKtide substrate phosphorylation level by autoradiographyMore data for this Ligand-Target Pair