Affinity DataKd: 3.10nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Average Binding Constant for TEK; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 46nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 57nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 240nMAssay Description:Average Binding Constant for TEK; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 270nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 280nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 300nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 300nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 300nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 310nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 310nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 370nMAssay Description:Binding affinity to human TIE2More data for this Ligand-Target Pair
Affinity DataKd: 395nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged TEK (unknown origin) (771 to 1124 residues) expressed in baculovirus infec...More data for this Ligand-Target Pair
Affinity DataKd: 408nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged TEK (unknown origin) (771 to 1124 residues) expressed in baculovirus infec...More data for this Ligand-Target Pair
Affinity DataKd: 440nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 450nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 450nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 450nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 450nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 450nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 450nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 630nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 630nMAssay Description:Binding affinity to TIE2More data for this Ligand-Target Pair
Affinity DataKd: 950nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 950nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 950nMAssay Description:Binding affinity to TIE2 (unknown origin) assessed as dissociation constant by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Binding constant for TIE2 kinase domainMore data for this Ligand-Target Pair