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Found 188 Enz. Inhib. hit(s) with Target = 'Taste receptor type 2 member 1'
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613033(CHEMBL5279691)
Affinity DataEC50:  72nMMore data for this Ligand-Target Pair
Ligand InfoPDB
In DepthDetails PDB3D3D Structure (crystal)
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613028(CHEMBL5285591)
Affinity DataEC50:  98nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613041(CHEMBL5275180)
Affinity DataEC50:  100nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613023(CHEMBL5273955)
Affinity DataEC50:  150nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613032(CHEMBL5274304)
Affinity DataEC50:  160nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613021(CHEMBL5277615)
Affinity DataEC50:  170nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613040(CHEMBL5280542)
Affinity DataEC50:  180nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613015(CHEMBL5279381)
Affinity DataEC50:  190nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50124575(CHEMBL3623735)
Affinity DataEC50:  190nMMore data for this Ligand-Target Pair
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613019(CHEMBL3088246)
Affinity DataEC50:  230nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613038(CHEMBL5277281)
Affinity DataEC50:  300nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613018(CHEMBL5278834)
Affinity DataEC50:  300nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613014(CHEMBL5278171)
Affinity DataEC50:  330nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613030(CHEMBL5274470)
Affinity DataEC50:  360nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613024(CHEMBL5278477)
Affinity DataEC50:  380nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613016(CHEMBL5275001)
Affinity DataEC50:  390nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613022(CHEMBL5289590)
Affinity DataEC50:  420nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM17636(2-{[3-(trifluoromethyl)phenyl]amino}benzoic acid |...)
Affinity DataEC50:  430nMMore data for this Ligand-Target Pair
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613036(CHEMBL5280688)
Affinity DataEC50:  540nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613034(CHEMBL5268924)
Affinity DataEC50:  640nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613020(CHEMBL5286379)
Affinity DataEC50:  640nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613025(CHEMBL5279341)
Affinity DataEC50:  670nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613037(CHEMBL5289980)
Affinity DataEC50:  750nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613012(CHEMBL5276181)
Affinity DataEC50:  930nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50385711(CHEMBL22815)
Affinity DataEC50:  950nMMore data for this Ligand-Target Pair
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613031(CHEMBL5265924)
Affinity DataEC50:  1.10E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613026(CHEMBL5268477)
Affinity DataEC50:  1.20E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613039(CHEMBL5280454)
Affinity DataEC50:  1.40E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613027(CHEMBL5274977)
Affinity DataEC50:  1.60E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613013(CHEMBL5285283)
Affinity DataEC50:  1.80E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613017(CHEMBL5288875)
Affinity DataEC50:  2.10E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613029(CHEMBL5265867)
Affinity DataEC50:  3.50E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50613035(CHEMBL5279932)
Affinity DataEC50:  6.80E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM50044849(CHEMBL3311308)
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at human TAS2R14 expressed in U2OS cells by Ga16gust44 Clone 7A FLIPR/summary (Abse5) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM211262(US9247759, 10-10)
Affinity DataEC50:  4.00E+4nMAssay Description:Agonist activity at TAS2R14 (unknown origin) by stably expressed cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 16(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50044849(CHEMBL3311308)
Affinity DataEC50: <5.01E+4nMAssay Description:Agonist activity at human TAS2R16 expressed in U2OS cells by summary (Abse5) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 1(Homo sapiens)
Firmenich

Curated by ChEMBL
LigandPNGBDBM211262(US9247759, 10-10)
Affinity DataEC50:  1.50E+5nMAssay Description:Agonist activity at TAS2R1 (unknown origin) by stably expressed cell-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM60947(BDBM50443972 | US9247759, compound C)
Affinity DataIC50:  200nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM60947(BDBM50443972 | US9247759, compound C)
Affinity DataIC50:  220nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM211081(US9247759, 5-2)
Affinity DataIC50:  590nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM211082(US9247759, 5-3)
Affinity DataIC50:  3.00E+3nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM211083(US9247759, 5-4)
Affinity DataIC50:  1.00E+4nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM211084(US9247759, 5-5)
Affinity DataIC50:  4.60E+3nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM211085(US9247759, 5-6)
Affinity DataIC50:  1.00E+4nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM211086(US9247759, 5-7)
Affinity DataIC50:  1.20E+4nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM211087(US9247759, 5-8)
Affinity DataIC50:  2.50E+3nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM211088(US9247759, 5-9)
Affinity DataIC50:  1.50E+4nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM211089(US9247759, 5-10 | US9247759, 5-69)
Affinity DataIC50:  1.97E+3nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM211090(US9247759, 5-11)
Affinity DataIC50:  14nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTaste receptor type 2 member 14(Homo sapiens (Human))TBA
LigandPNGBDBM211093(US9247759, 5-14)
Affinity DataIC50:  1.88E+3nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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