Affinity DataKd: 1.20nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.90nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 5nMAssay Description:Binding affinity to human EPHA4More data for this Ligand-Target Pair
Affinity DataKd: 8.30nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Binding affinity to 6His-tagged EphA4 C204A mutant (29 to 104 residues) (unknown origin) expressed in Escherichia coli Origami 2 (DE3) by isothermal ...More data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Binding affinity to 6His-tagged EphA4 C204A mutant (29 to 104 residues) (unknown origin) expressed in Escherichia coli Origami 2 (DE3) by isothermal ...More data for this Ligand-Target Pair
Affinity DataKd: 30nMAssay Description:Binding affinity to 6His-tagged EphA4 C204A mutant (29 to 104 residues) (unknown origin) expressed in Escherichia coli Origami 2 (DE3) by isothermal ...More data for this Ligand-Target Pair
Affinity DataKd: 45nMAssay Description:Binding affinity to 6His-tagged EphA4 C204A mutant (29 to 104 residues) (unknown origin) expressed in Escherichia coli Origami 2 (DE3) by isothermal ...More data for this Ligand-Target Pair
Affinity DataKd: 60nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
TargetEphrin type-A receptor 4 [29-209,M164A](Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute
Sanford Burnham Prebys Medical Discovery Institute
Affinity DataKd: 62nMpH: 6.5 T: 2°CAssay Description:The purified EphA proteins (EphA4-LBD, EphA3-LBD, and EphA2-LBD) were dissolved in 50 mM potassium phosphate buffer (pH 6.5) containing 100 mM NaCl. ...More data for this Ligand-Target Pair
Affinity DataKd: 77nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 94nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 106nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 106nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 113nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 132nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 144nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 191nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 196nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 258nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 270nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
TargetEphrin type-A receptor 4 [29-209,I159A](Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute
Sanford Burnham Prebys Medical Discovery Institute
Affinity DataKd: 290nMpH: 6.5 T: 2°CAssay Description:The purified EphA proteins (EphA4-LBD, EphA3-LBD, and EphA2-LBD) were dissolved in 50 mM potassium phosphate buffer (pH 6.5) containing 100 mM NaCl. ...More data for this Ligand-Target Pair
Affinity DataKd: 307nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 310nMAssay Description:Average Binding Constant for EPHA4; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 330nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
TargetEphrin type-A receptor 4 [29-209,D61G,E62G](Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute
Sanford Burnham Prebys Medical Discovery Institute
Affinity DataKd: 340nMpH: 6.5 T: 2°CAssay Description:The purified EphA proteins (EphA4-LBD, EphA3-LBD, and EphA2-LBD) were dissolved in 50 mM potassium phosphate buffer (pH 6.5) containing 100 mM NaCl. ...More data for this Ligand-Target Pair
TargetEphrin type-A receptor 4 [29-209,M60A](Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute
Sanford Burnham Prebys Medical Discovery Institute
Affinity DataKd: 350nMpH: 6.5 T: 2°CAssay Description:The purified EphA proteins (EphA4-LBD, EphA3-LBD, and EphA2-LBD) were dissolved in 50 mM potassium phosphate buffer (pH 6.5) containing 100 mM NaCl. ...More data for this Ligand-Target Pair
Affinity DataKd: 352nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 360nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 362nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 370nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 400nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 400nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 400nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 400nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 420nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 420nMAssay Description:Binding affinity to EphA4 ligand binding domain (unknown origin) by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 420nMAssay Description:Binding constant for EPHA4 kinase domainMore data for this Ligand-Target Pair
TargetEphrin type-A receptor 4 [29-209](Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute
Sanford Burnham Prebys Medical Discovery Institute
Affinity DataKd: 420nMpH: 6.5 T: 2°CAssay Description:The purified EphA proteins (EphA4-LBD, EphA3-LBD, and EphA2-LBD) were dissolved in 50 mM potassium phosphate buffer (pH 6.5) containing 100 mM NaCl. ...More data for this Ligand-Target Pair
Affinity DataKd: 420nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 437nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 444nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair
Affinity DataKd: 459nMAssay Description:Binding affinity to N-terminal His tagged EphA4 LBD (unknown origin) (29 to 209 residues) expressed in Rosetta-Gami B(DE3) cells by isothermal titrat...More data for this Ligand-Target Pair