Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) for PDB: 2QT9
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221979((2S,3S)-2-((1r,4S)-4-([1,2,4]triazolo[1,5-a]pyridi...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221979((2S,3S)-2-((1r,4S)-4-([1,2,4]triazolo[1,5-a]pyridi...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50221979((2S,3S)-2-((1r,4S)-4-([1,2,4]triazolo[1,5-a]pyridi...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human DPP4 in presence of 50 % human serumMore data for this Ligand-Target Pair