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Found 2 Enz. Inhib. hit(s) for PDB: 4F1L
TargetProtein mono-ADP-ribosyltransferase PARP14(Homo sapiens (Human))
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM50397960(CHEMBL2179989)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of hexahistidine-tagged human recombinant ARTD8 catalytic domain (1611 to 1801 amino acids) expressed in Escherichia coli BL21(DE3) assess...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14(Homo sapiens (Human))
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM50397960(CHEMBL2179989)
Affinity DataKd:  7.60E+3nMAssay Description:Binding affinity at human recombinant ARTD8 expressed in Escherichia coli BL21 (DE3) R3 pRARE cells by isothermal titration calorimetryMore data for this Ligand-Target Pair