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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) for PDB:
5I88
Target
Bromodomain-containing protein 4 [42-168]
(Homo sapiens (Human))
Genentech
US Patent
Ligand
BDBM321357
(3-(6-but-2-enyl-7-oxo-1H-pyrrolo[2,3-c]pyridin-4-y...)
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Affinity Data
IC50: 330nM
Assay Description:
His/Flag epitope tagged BRD4 BD142-168 was cloned, expressed, and purified to homogeneity. BRD4 binding and inhibition was assessed by monitoring the...
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Target Info
PDB
UniProtKB/SwissProt
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Ligand Info
PC cid
PC sid
PDB
In Depth
Details
US Patent
PDB
3D Structure (crystal)
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