Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 50013028
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125604(1-[9-Benzyl-2-(2-fluoro-phenyl)-9H-purin-6-yl]-1-(...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125605(1-(2,6-Difluoro-phenyl)-1-[2-(2,4-difluoro-phenyl)...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125600(1-[2-(2-Chloro-phenyl)-9-methyl-9H-purin-6-yl]-1-(...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125606(1-(2,6-Difluoro-phenyl)-1-[2-(2-fluoro-phenyl)-9-m...)
Affinity DataIC50:  36nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125597(1-(2,6-Difluoro-phenyl)-1-[9-(2-dimethylamino-ethy...)
Affinity DataIC50:  82nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125601(1-(2-Chloro-phenyl)-1-[2-(4-fluoro-2-methyl-phenyl...)
Affinity DataIC50:  123nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125602(1-(2,6-Difluoro-phenyl)-1-[2-(4-fluoro-2-methyl-ph...)
Affinity DataIC50:  128nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125589(1-(2,6-Difluoro-phenyl)-1-(9-methyl-2-o-tolyl-9H-p...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125598(1-[2-(4-Fluoro-2-methyl-phenyl)-9-methyl-9H-purin-...)
Affinity DataIC50:  163nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125592(1-(2,6-Difluoro-phenyl)-1-(9-methyl-2-m-tolyl-9H-p...)
Affinity DataIC50:  350nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125599(1-(2,6-Difluoro-phenyl)-1-(9-methyl-2-phenyl-9H-pu...)
Affinity DataIC50:  510nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125607(1-[2-(3-Chloro-phenyl)-9-methyl-9H-purin-6-yl]-1-(...)
Affinity DataIC50:  550nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125596(1-(2,6-Difluoro-phenyl)-1-[2-(4-fluoro-phenyl)-9-m...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125594(1-[2-(4-Fluoro-2-methyl-phenyl)-9-methyl-9H-purin-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125590(1-(2,6-Difluoro-phenyl)-1-(9-methyl-2-p-tolyl-9H-p...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125595(1-(2,6-Difluoro-phenyl)-1-[2-(3-fluoro-phenyl)-9-m...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125608(1-(4-Chloro-phenyl)-1-[2-(4-fluoro-2-methyl-phenyl...)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125603(1-[2-(4-Fluoro-2-methyl-phenyl)-9-methyl-9H-purin-...)
Affinity DataIC50: >1.67E+4nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125593(1-(2,6-Difluoro-phenyl)-1-[2-(3,5-difluoro-phenyl)...)
Affinity DataIC50: >1.67E+4nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50125591(1-[2-(4-Fluoro-2-methyl-phenyl)-9-methyl-9H-purin-...)
Affinity DataIC50: >1.67E+4nMAssay Description:Inhibition of human MAP p38-alpha kinase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed