Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with all data for entry = 50017344
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50180789(1,2-bis(7-methyl-[1,2,4]triazolo[4,3-a]pyridin-3-y...)
Affinity DataIC50:  400nMAssay Description:Inhibition of recombinant CpG methylase M.SssIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50180790(2-(1,3-dioxoisoindolin-2-yl)-3-(1H-indol-3-yl)prop...)
Affinity DataIC50:  600nMAssay Description:Inhibition of recombinant CpG methylase M.SssIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50180790(2-(1,3-dioxoisoindolin-2-yl)-3-(1H-indol-3-yl)prop...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory activity against DNA methyl transferase in leukemic NALM6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50180789(1,2-bis(7-methyl-[1,2,4]triazolo[4,3-a]pyridin-3-y...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibitory activity against DNA methyl transferase in leukemic NALM6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed