Compile Data Set for Download or QSAR
maximum 50k data
Found 40 Enz. Inhib. hit(s) with all data for entry = 50003875
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476896(CHEMBL232576)
Affinity DataIC50:  2nMAssay Description:Inhibition of HIV1 reverse transcriptase by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476895(CHEMBL232379)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of HIV1 reverse transcriptase by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476903(CHEMBL230188)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of HIV1 reverse transcriptase by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476898(CHEMBL232377)
Affinity DataIC50:  5nMAssay Description:Inhibition of HIV1 reverse transcriptase by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476897(CHEMBL232178)
Affinity DataIC50:  5nMAssay Description:Inhibition of HIV1 reverse transcriptase by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476904(CHEMBL232575)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of HIV1 reverse transcriptase by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476885(CHEMBL231030)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of HIV1 reverse transcriptase by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476894(CHEMBL230187)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of HIV1 reverse transcriptase by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476899(CHEMBL232963)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476896(CHEMBL232576)
Affinity DataIC50:  8.90nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM27606(2-{[1-(naphthalen-1-yl)-1H-1,2,3,4-tetrazol-5-yl]s...)
Affinity DataIC50:  9.5nMAssay Description:Inhibition of HIV1 reverse transcriptase by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476893(CHEMBL393190)
Affinity DataIC50:  10nMAssay Description:Inhibition of HIV1 reverse transcriptase by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476909(CHEMBL232378)
Affinity DataIC50:  10nMAssay Description:Inhibition of HIV1 reverse transcriptase by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476904(CHEMBL232575)
Affinity DataIC50:  12nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476892(CHEMBL391298)
Affinity DataIC50:  16nMAssay Description:Inhibition of HIV1 reverse transcriptase by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476891(CHEMBL233167)
Affinity DataIC50:  17nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476889(CHEMBL232765)
Affinity DataIC50:  17nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476905(CHEMBL231980)
Affinity DataIC50:  19nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476887(CHEMBL232764)
Affinity DataIC50:  20nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476906(CHEMBL393423)
Affinity DataIC50:  23nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476888(CHEMBL231777)
Affinity DataIC50:  23nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476902(CHEMBL231981)
Affinity DataIC50:  26nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476903(CHEMBL230188)
Affinity DataIC50:  26nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM27607(4-[3-chloro-4-(2-{[1-(2-chloro-4-cyclopropylphenyl...)
Affinity DataIC50:  28nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476886(CHEMBL232962)
Affinity DataIC50:  30nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476901(CHEMBL393816)
Affinity DataIC50:  32nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476893(CHEMBL393190)
Affinity DataIC50:  33nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476885(CHEMBL231030)
Affinity DataIC50:  36nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476900(CHEMBL232961)
Affinity DataIC50:  38nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476895(CHEMBL232379)
Affinity DataIC50:  38nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476910(CHEMBL393990)
Affinity DataIC50:  43nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476907(CHEMBL393191)
Affinity DataIC50:  44nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476898(CHEMBL232377)
Affinity DataIC50:  45nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476890(CHEMBL393422)
Affinity DataIC50:  47nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476897(CHEMBL232178)
Affinity DataIC50:  66nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476908(CHEMBL232766)
Affinity DataIC50:  80nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476894(CHEMBL230187)
Affinity DataIC50:  94nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476909(CHEMBL232378)
Affinity DataIC50:  150nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM50476892(CHEMBL391298)
Affinity DataIC50:  151nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada)

Curated by ChEMBL
LigandPNGBDBM27606(2-{[1-(naphthalen-1-yl)-1H-1,2,3,4-tetrazol-5-yl]s...)
Affinity DataIC50:  766nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed