Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50025628
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50264830(CHEMBL492052 | N-(3-Benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in Wistar rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50264830(CHEMBL492052 | N-(3-Benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50264830(CHEMBL492052 | N-(3-Benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]CGS21680 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50265409(CHEMBL496985 | N6-[(4-Amino)-phenyl]-9-benzyl-2-ph...)
Affinity DataKi:  294nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in Wistar rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50265409(CHEMBL496985 | N6-[(4-Amino)-phenyl]-9-benzyl-2-ph...)
Affinity DataKi:  396nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50265408(CHEMBL496984 | N6-[(4-Nitro)-phenyl]-9-benzyl-2-ph...)
Affinity DataKi:  571nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in Wistar rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50265408(CHEMBL496984 | N6-[(4-Nitro)-phenyl]-9-benzyl-2-ph...)
Affinity DataKi:  699nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50264830(CHEMBL492052 | N-(3-Benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50265408(CHEMBL496984 | N6-[(4-Nitro)-phenyl]-9-benzyl-2-ph...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50265409(CHEMBL496985 | N6-[(4-Amino)-phenyl]-9-benzyl-2-ph...)
Affinity DataKi:  4.17E+3nMAssay Description:Displacement of [3H]CGS21680 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50264885(1-[4-(9-Benzyl-2-phenyl-9H-purin-6-ylamino)-phenyl...)
Affinity DataKi:  5.61E+3nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50265409(CHEMBL496985 | N6-[(4-Amino)-phenyl]-9-benzyl-2-ph...)
Affinity DataKi:  5.74E+3nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50264830(CHEMBL492052 | N-(3-Benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataEC50:  750nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50264830(CHEMBL492052 | N-(3-Benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataEC50:  9.74E+3nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50264831(1-[4-(3-Benzyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]-...)
Affinity DataEC50:  1.60E+4nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50264831(1-[4-(3-Benzyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]-...)
Affinity DataEC50:  9.95E+3nMAssay Description:Displacement of [3H]CGS21680 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed