Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50000847
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM22885(3-[(2S)-1-(1H-imidazol-5-yl)propan-2-yl]-2-(2-{[(5...)
Affinity DataKi:  40nMAssay Description:Evaluated for antagonistic activity at histamine H3 receptor in rat cerebral cortex and is represented as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM85411(GT 2174)
Affinity DataKi:  50nMAssay Description:Evaluated for antagonist activity against histamine H3 receptor and is represented as -log Ki.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM22886(3-[(2R)-1-(1H-imidazol-5-yl)propan-2-yl]-2-(2-{[(5...)
Affinity DataKi:  60nMAssay Description:Evaluated for antagonistic activity at histamine H3 receptor in rat cerebral cortex and is represented as Ki.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50406098(CHEMBL12494)
Affinity DataKi:  79nMAssay Description:Evaluated for antagonist activity against Histamine H3 receptor and represented as KB.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50406100(CHEMBL12459)
Affinity DataKi:  200nMAssay Description:Evaluated for antagonist activity against Histamine H3 receptor and represented as KB.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50406095(CHEMBL275090)
Affinity DataKi:  631nMAssay Description:Evaluated for antagonist activity against histamine H3 receptor and is represented as -log Ki.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50406101(CHEMBL12550)
Affinity DataKi:  631nMAssay Description:Evaluated for antagonist activity against Histamine H3 receptor and represented as KB.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50406099(CHEMBL416338)
Affinity DataKi:  1.00E+3nMAssay Description:Evaluated for antagonist activity against histamine H3 receptor and is represented as -log Ki.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50406096(CHEMBL12025)
Affinity DataKi:  1.00E+3nMAssay Description:Evaluated for antagonist activity against Histamine H3 receptor and represented as KB.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50406093(CHEMBL276903)
Affinity DataKi:  1.00E+3nMAssay Description:Evaluated for antagonist activity against Histamine H3 receptor and represented as KB.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50406097(CHEMBL12551)
Affinity DataKi:  1.00E+3nMAssay Description:Evaluated for antagonist activity against histamine H3 receptor and is represented as -log Ki.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed