TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 810nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 870nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair