TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Affinity DataEC50: 50.1nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 2.51E+3nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 1.58E+3nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 3.16E+3nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 794nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 631nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 1.58E+4nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 501nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 63.1nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair